BARC/PUB/2012/1353

 
 

An enantiodivergent and formal synthesis of paroxetine enantiomers by asymmetric desymmetrization of 3-(4-fluorophenyl)glutaric anhydride with a chiral SuperQuat oxazolidin-2-one

 
     
 
Author(s)

Chaubey, N. R.; Ghosh, S. K.
(BOD)

Source

Tetrahedron-Asymmetry, 2012. Vol. 23: pp. 1206-1212

ABSTRACT

The asymmetric desymmetrization of 3-(4-fluorophenyl)glutaric anhydride 9 with lithiated chiral oxazolidin-2-one 8 has been studied. The desymmetrized product was formed with >90% de and converted into known intermediates for both (+)- and (-)-paroxetines.

 
 
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